SCHEMBL5990167

SCHEMBL5990167

COc1ccc(OC(F)(F)F)cc1Oc1ccccc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.49
SCN8A Q9UQD0 1/20 0.48
SCN10A Q9Y5Y9 1/20 0.48
BCAT1 P54687 2/20 0.44
BCAT2 O15382 1/20 0.44
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
GRIN2B Q13224 2/20 0.42
ALPL P05186 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
BRAF P15056 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5990326 0.84 SCN8A (0.49) ARSCN8ASCN10AHTTSLC6A2
SCHEMBL12180463 0.81 GPR3 (0.44) GRIN2BCA12CA1CA2CA7
SCHEMBL12422184 0.81 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL13680420 0.79 SLC6A4 (0.58) ARSCN8ASCN10ABCAT1BCAT2
SCHEMBL8302095 0.77 GPR3 (0.44) ALPLCA12CA1CA2CA7
SCHEMBL8014909 0.75 CA1 (0.62) ARALDH1A1MAPK1HTTL3MBTL1
SCHEMBL5990449 0.74 AR (0.50) ARHTTCA12CA1CA2
SCHEMBL23957964 0.73 AR (0.56) ARBCAT1BCAT2ALDH1A1MAPK1
SCHEMBL20650170 0.73 GPR3 (0.46) MAPK1GRIN2BSLC6A2SLC6A3
SCHEMBL3033181 0.73 RUNX1 (0.42) ALDH1A1GRIN2BALPLCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060257987-A1 Ppar modulators ELI LILLY AND COMPANY 2006-11-16 US disclosed
EP-1660428-A1 PPAR MODULATORS ELI LILLY AND COMPANY (US) 2006-05-31 EP disclosed
WO-2005019151-A1 PPAR MODULATORS ELI LILLY AND COMPANY (US) 2005-03-03 WO disclosed