SCHEMBL5994352

SCHEMBL5994352

COc1ccc2[nH]nc(C(=O)NC3CN4CCC3CC4)c2c1

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 2/20 0.70
CHRNA7 P36544 1/20 0.70
GSK3B P49841 16/20 0.58
HTR3E A5X5Y0 1/20 0.52
HTR3B O95264 1/20 0.52
HTR3D Q70Z44 1/20 0.52
HTR3C Q8WXA8 1/20 0.52
CDK2 P24941 1/20 0.50
CDK16 Q00536 1/20 0.50
DYRK1A Q13627 1/20 0.50
ROCK1 Q13464 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1964521 1.00 HTR3A (0.70) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL1964257 1.00 HTR3A (0.70) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL1963670 0.92 CHRNA7 (0.70) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL1963239 0.92 CHRNA7 (0.70) HTR3ACHRNA7GSK3BHTR3EHTR3B
Hydrochloric Acid SCHEMBL1963923 0.91 CHRNA7 (0.69) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL5995368 0.88 CHRNA7 (0.67) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL1963576 0.88 CHRNA7 (0.67) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL1963569 0.88 CHRNA7 (0.67) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL1965364 0.88 CHRNA7 (0.67) HTR3ACHRNA7GSK3BHTR3EHTR3B
SCHEMBL2787737 0.88 CHRNA7 (0.64) HTR3ACHRNA7GSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735306-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF Memory Pharmaceuticals Corporation (US) 2006-12-27 EP disclosed
WO-2005092890-A2 INDAZOLES, BENZOTHIAZOLES, BENZOISOTHIAZOLES, BENZISOXAZOLES, AND PREPARATION AND USES THEREOF MEMORY PHARMACEUTICALS CORPORATION (US) 2005-10-06 WO disclosed