SCHEMBL5994928

SCHEMBL5994928

CNC(=O)c1ccccc1Sc1c[nH]c2cccc(C)c12.CNC(=O)c1ccccc1Sc1c[nH]c2cccc(Cl)c12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR4A2 P43354 1/20 0.45
IDO1 P14902 2/20 0.44
SLC6A3 Q01959 3/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
MAPT P10636 1/20 0.40
PTGER3 P43115 2/20 0.39
NPC1 O15118 1/20 0.39
AR P10275 1/20 0.38
GPR84 Q9NQS5 2/20 0.37
ITGB2 P05107 1/20 0.37
ICAM1 P05362 1/20 0.37
ITGAL P20701 1/20 0.37
PLK4 O00444 2/20 0.37
AURKA O14965 2/20 0.37
MAP4K4 O95819 2/20 0.37
PAK4 O96013 2/20 0.37
ABL1 P00519 2/20 0.37
LCK P06239 2/20 0.37
CSF1R P07333 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399253 0.95 NR4A2 (0.49) NR4A2IDO1SLC6A3SLC6A2SLC6A4
SCHEMBL1399410 0.93 SLC6A3 (0.49) NR4A2IDO1SLC6A3SLC6A2SLC6A4
SCHEMBL1399366 0.79 ALDH1A1 (0.55) NR4A2IDO1SLC6A4MAPTPTGER3
SCHEMBL1399364 0.77 GFER (0.52) NR4A2IDO1SLC6A3SLC6A2SLC6A4
SCHEMBL1399287 0.76 HPGD (0.48) IDO1SLC6A4MAPTNPC1GPR84
SCHEMBL1399315 0.72 IFNAR1 (0.51) NR4A2IDO1SLC6A3SLC6A2SLC6A4
SCHEMBL5908998 0.71 IDO1 (0.40) NR4A2IDO1SLC6A2SLC6A4PTGER3
SCHEMBL4385853 0.71 TAAR1 (0.50) NR4A2IDO1SLC6A2SLC6A4PTGER3
SCHEMBL1399293 0.70 IFNAR1 (0.54) IDO1SLC6A3SLC6A2SLC6A4MAPT
SCHEMBL4389000 0.69 IDO1 (0.46) NR4A2IDO1SLC6A2SLC6A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701940-A1 2-(1H-INDOLYLSULFANYL)-BENZYL AMINE DERIVATIVES AS SSRI H.Lundbeck A/S (DK) 2006-09-20 EP disclosed
EP-1654247-A1 ALKYNYL ARYL CARBOXAMIDES Applied Research Systems ARS Holding N.V. (AN) 2006-05-10 EP disclosed
WO-2005061455-A1 2-(1H-INDOLYLSULFANYL)-BENZYL AMINE DERIVATIVES AS SSRI H. LUNDBECK A/S (DK) 2005-07-07 WO disclosed
WO-2005012280-A1 ALKYNYL ARYL CARBOXAMIDES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2005-02-10 WO disclosed