SCHEMBL5998293

SCHEMBL5998293

COc1ccc(Cl)c(C(=O)Nc2cnc(Nc3ccc(C(=O)O)nc3)nc2)c1

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 1/20 0.56
P4HTM Q9NXG6 1/20 0.53
BTK Q06187 2/20 0.49
BLK P51451 1/20 0.49
RORC P51449 1/20 0.49
MAPT P10636 1/20 0.48
LCK P06239 1/20 0.48
CSF1R P07333 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5998110 0.87 P4HTM (0.48) P4HTMBTK
SCHEMBL5997052 0.84 CSF1R (0.64) TYK2MAPTCSF1R
SCHEMBL5997760 0.83 TYK2 (0.51) TYK2BTKBLKMAPTCSF1R
SCHEMBL15100315 0.81 TYK2 (0.70) TYK2MAPTCSF1R
SCHEMBL5996482 0.81 SRC (0.51) TYK2BTKBLKMAPTLCK
SCHEMBL5996063 0.77 PDGFRB (0.56) TYK2BTKBLKLCK
SCHEMBL2324574 0.76 RORC (0.57) P4HTMRORCMAPT
SCHEMBL15561708 0.76
SCHEMBL5281904 0.75 LCK (0.58) TYK2P4HTMRORCLCK
SCHEMBL2495621 0.75 BTK (0.75) BTKBLKLCKCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060247250-A1 Pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2006-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060247250-A1 Pyrimidine inhibitors of kinases DTYMK, SRC, DCK TYK2 5/4885P4HTM 3856/4885BTK 19/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.