SCHEMBL5998680

SCHEMBL5998680

CCOC(=O)C(CN1C(=O)c2ccc(Br)cc2C1=O)C(C)=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
PIN1 Q13526 1/20 0.45
PIN4 Q9Y237 1/20 0.45
SMAD3 P84022 2/20 0.44
APAF1 O14727 1/20 0.44
KDM1A O60341 1/20 0.42
CUL4A Q13619 1/20 0.41
ESR1 P03372 2/20 0.40
GABRA1 P14867 2/20 0.40
GABRG2 P18507 2/20 0.40
GABRB3 P28472 2/20 0.40
GABRA5 P31644 2/20 0.40
GABRA3 P34903 2/20 0.40
GABRA2 P47869 2/20 0.40
GABRA6 Q16445 2/20 0.40
ESR2 Q92731 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
TDP2 O95551 1/20 0.39
POLB P06746 3/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5998277 0.88 ALDH1A1 (0.56) ALDH1A1SMAD3APAF1KDM1ACUL4A
SCHEMBL5996615 0.87 PIN1 (0.47) ALDH1A1PIN1PIN4POLBMAPK1
SCHEMBL5995992 0.85 PIN1 (0.45) ALDH1A1PIN1PIN4GABRA1GABRG2
SCHEMBL5998506 0.85 PIN1 (0.45) ALDH1A1PIN1PIN4GABRA1GABRG2
SCHEMBL5998387 0.84 ALDH1A1 (0.49) ALDH1A1PIN1PIN4MEN1KMT2A
SCHEMBL5998140 0.82 CA9 (0.43) ALDH1A1PIN1PIN4NPC1
SCHEMBL5998787 0.81 PIN1 (0.42) ALDH1A1PIN1PIN4MAPK1MEN1
SCHEMBL5998421 0.81 RPS6KA2 (0.50) ALDH1A1MEN1KMT2A
SCHEMBL5998692 0.79 ALDH1A1 (0.47) ALDH1A1PIN1PIN4SMAD3APAF1
SCHEMBL522944 0.79 PIN1 (0.68) ALDH1A1PIN1PIN4RXFP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7094908-B2 Reduction of carbonyl compounds using the carbonyl reductase of Kluyveromyces marxianus KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2006-08-22 US disclosed
US-20030139464-A1 Reduction of carbonyl compounds using the carbonyl reductase of kluyveromyces marxianus KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY 2003-07-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030139464-A1 Reduction of carbonyl compounds using the carbonyl reductase of kluyveromyces marxianus CBR1, CBR3, DCXR ALDH1A1 216/4885PIN1 1143/4885PIN4 695/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.