SCHEMBL6002906

SCHEMBL6002906

[CH2]COCCc1ccc2sccc2c1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.54
CYP2A6 P11509 2/20 0.53
PDE10A Q9Y233 1/20 0.38
DYRK1A Q13627 1/20 0.35
PTPRC P08575 1/20 0.35
PTPN6 P29350 1/20 0.35
PTPN11 Q06124 1/20 0.35
PTPN22 Q9Y2R2 1/20 0.35
CA12 O43570 4/20 0.35
CA2 P00918 4/20 0.35
CTNNB1 P35222 1/20 0.34
WNT3A P56704 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
TPSAB1 Q15661 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13873189 0.84 SIGMAR1 (0.57) SIGMAR1CYP2A6PDE10ADYRK1APTPRC
SCHEMBL3816500 0.83 SIGMAR1 (0.56) SIGMAR1CYP2A6PDE10ADYRK1APTPRC
SCHEMBL3813009 0.83 SIGMAR1 (0.60) SIGMAR1CYP2A6PDE10ADYRK1APTPRC
SCHEMBL2091182 0.81 CYP2A6 (0.61) SIGMAR1CYP2A6PDE10ADYRK1APTPRC
SCHEMBL3810261 0.81 SIGMAR1 (0.49) SIGMAR1CYP2A6PDE10ACA12CA2
SCHEMBL52071 0.80 SIGMAR1 (0.60) SIGMAR1CYP2A6PDE10ACA12CA2
SCHEMBL10368304 0.80 SIGMAR1 (0.51) SIGMAR1CYP2A6PDE10APTPRCPTPN6
SCHEMBL3816494 0.80 SIGMAR1 (0.51) SIGMAR1CYP2A6PDE10ADYRK1APTPRC
SCHEMBL52010 0.80 SIGMAR1 (0.51) SIGMAR1CYP2A6PDE10ADYRK1APTPRC
SCHEMBL47966 0.80 SIGMAR1 (0.60) SIGMAR1CYP2A6PDE10ADYRK1APTPRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed