SCHEMBL6004442

SCHEMBL6004442

Br[Mg]c1ccccc1.Nc1c(Cl)cccc1C(=O)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
GAA P10253 1/20 0.46
MAPK14 Q16539 2/20 0.46
LMNA P02545 3/20 0.45
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 1/20 0.45
USP2 O75604 1/20 0.45
GLA P06280 1/20 0.45
KMT2A Q03164 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ADORA1 P30542 2/20 0.41
AKR1C3 P42330 1/20 0.41
POLB P06746 2/20 0.41
ABCB11 O95342 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NR4A1 P22736 1/20 0.40
ALOX15 P16050 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31366601 0.88 GAA (0.58) MAPTGAAMAPK14LMNAALDH1A1
SCHEMBL1569037 0.88 GAA (0.58) MAPTGAAMAPK14LMNAALDH1A1
SCHEMBL11320848 0.77 NR4A1 (0.56) MAPTMAPK14LMNAALDH1A1MEN1
SCHEMBL10931534 0.75 MAPT (0.53) MAPTGAAMAPK14LMNAALDH1A1
SCHEMBL342695 0.74 TYK2 (0.49) MAPTGAAMAPK14LMNAALDH1A1
SCHEMBL15628209 0.74 ALOX15 (0.54) MAPTLMNAALDH1A1MEN1KMT2A
SCHEMBL11320349 0.74 AKR1C3 (0.53) MAPTGAALMNAALDH1A1KMT2A
SCHEMBL8956729 0.74 KMT2A (0.44) MAPTMAPK14LMNAALDH1A1MEN1
SCHEMBL35142 0.73 HSD17B1 (0.49) ALDH1A1POLB
SCHEMBL49873 0.72 KMT2A (0.65) MAPTGAALMNAALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1641781-A2 BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2006-04-05 EP disclosed
WO-2005000807-A2 BENZODIAZEPINE CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2005-01-06 WO disclosed