SCHEMBL6004777

SCHEMBL6004777

O=C(Cl)c1ccc(OCCC2CCCCCN2)cc1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.54
LTA4H P09960 12/20 0.46
HRH2 P25021 1/20 0.45
HRH1 P35367 1/20 0.45
AURKB Q96GD4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5706378 0.99 CHEK2 (0.55) CHEK2LTA4HHRH2HRH1AURKB
Hydrochloric Acid SCHEMBL6560096 0.97 CHEK2 (0.54) CHEK2LTA4HHRH2HRH1AURKB
SCHEMBL3866051 0.87 CHEK2 (0.56) CHEK2LTA4HHRH2HRH1
Hydrochloric Acid SCHEMBL6561583 0.86 CHEK2 (0.55) CHEK2LTA4HHRH2HRH1
SCHEMBL7447377 0.85 LTA4H (0.56) CHEK2LTA4HHRH2HRH1AURKB
SCHEMBL6560708 0.84 MAPT (0.56) CHEK2LTA4HHRH2HRH1
SCHEMBL7335065 0.84 LTA4H (0.54) CHEK2LTA4H
SCHEMBL6053346 0.84 CHEK2 (0.58) CHEK2LTA4HHRH2HRH1
Hydrochloric Acid SCHEMBL7328923 0.82 LTA4H (0.53) CHEK2LTA4H
SCHEMBL6005460 0.82 LTA4H (0.49) CHEK2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1709021-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS ELI LILLY AND COMPANY (US) 2006-10-11 EP disclosed
WO-2005073204-A1 SELECTIVE ESTROGEN RECEPTOR MODULATORS FOR THE TREATMENT OF VASOMOTOR SYMPTOMS ELI LILLY AND COMPANY (US) 2005-08-11 WO disclosed