SCHEMBL6005902

SCHEMBL6005902

O=Nc1nccc2nc(-c3ccco3)nn12

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.48
ADORA1 P30542 5/20 0.44
ADORA2B P29275 2/20 0.44
ADORA3 P0DMS8 3/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TDP1 Q9NUW8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3548138 0.82 ADORA2A (0.63) ADORA2AADORA1ADORA2BADORA3
SCHEMBL30507661 0.72 KDM4E (0.46) ADORA2AADORA1ADORA2BADORA3KDM4E
SCHEMBL7152951 0.71 ADORA2A (0.56) ADORA2AADORA1ADORA2BADORA3
SCHEMBL5653322 0.69 ADORA2A (0.71) ADORA2AADORA1ADORA2B
SCHEMBL13979684 0.68 ADORA2A (0.43) ADORA2AADORA1ADORA2BADORA3KDM4E
SCHEMBL6047213 0.68 ADORA2A (0.82) ADORA2A
SCHEMBL9429556 0.67 RAB9A (0.46) ADORA2AADORA1KDM4EALDH1A1TDP1
SCHEMBL6047267 0.67 ADORA2A (0.74) ADORA2A
SCHEMBL30153455 0.67 ADORA2A (0.61) ADORA2AADORA1ADORA2BADORA3KDM4E
SCHEMBL6047223 0.67 ADORA2A (0.64) ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633756-A2 A2A ADENOSINE RECEPTOR ANTAGONISTS Biogen Idec MA Inc. (US) 2006-03-15 EP disclosed
WO-2004092173-A2 A2A ADENOSINE RECEPTOR ANTAGONISTS BIOGEN IDEC MA INC. (US) 2004-10-28 WO disclosed