SCHEMBL6008973

SCHEMBL6008973

CCCCC1N(CC2CCCCC2)C(=O)OC12CCN(C1CCN(C(=O)c3cscc3OC)CC1)CC2

nearest known ligand 0.71

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.71
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
TSHR P16473 1/20 0.36
HTT P42858 1/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6009082 0.86 CCR5 (0.81) CCR5CNR1
SCHEMBL6008167 0.84 CCR5 (0.72) CCR5
SCHEMBL6006898 0.82 CCR5 (0.80) CCR5
SCHEMBL6007387 0.82 CCR5 (0.84) CCR5KDM4EALDH1A1
SCHEMBL6006856 0.82 CCR5 (0.74) CCR5
SCHEMBL6005547 0.82 CCR5 (0.81) CCR5KDM4EALDH1A1
SCHEMBL6009109 0.81 CCR5 (0.88) CCR5CNR1
SCHEMBL6008971 0.81 CCR5 (0.75) CCR5
SCHEMBL6006576 0.81 CCR5 (0.75) CCR5KDM4E
SCHEMBL6005631 0.81 CCR5 (0.70) CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1716156-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2006-11-02 EP claimed
WO-2005075484-A2 CHEMOKINE CCR5 RECEPTOR MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-08-18 WO claimed