SCHEMBL6009016

SCHEMBL6009016

C[C@H]1COc2c(N3CC4CC4(N)C3)c(F)c(N)c3c(=O)c(C(=O)O)cn1c23

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 10/20 0.52
TOP2A P11388 3/20 0.48
TOP2B Q02880 3/20 0.48
AADAT Q8N5Z0 2/20 0.48
POLB P06746 2/20 0.48
CACNA1F O60840 1/20 0.48
MAPK1 P28482 1/20 0.48
CACNA1D Q01668 1/20 0.48
KCNH2 Q12809 1/20 0.48
CACNA1S Q13698 1/20 0.48
CACNA1C Q13936 1/20 0.48
KDM4E B2RXH2 4/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
HSD17B10 Q99714 2/20 0.47
ALB P02768 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
TUBB4A P04350 1/20 0.46
TUBB P07437 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6009397 0.84 AADAT (0.69) TOP2ATOP2BAADATPOLBKCNH2
SCHEMBL6204362 0.83 GSK3B (0.51) GSK3BTOP2ATOP2BAADATPOLB
SCHEMBL6204357 0.83 GSK3B (0.51) GSK3BTOP2ATOP2BAADATPOLB
SCHEMBL6635916 0.83 GSK3B (0.49) GSK3BTOP2ATOP2BAADATPOLB
SCHEMBL10684313 0.82 KDM4E (0.68) GSK3BTOP2ATOP2BAADATPOLB
SCHEMBL29391130 0.82 KDM4E (0.68) GSK3BTOP2ATOP2BAADATPOLB
SCHEMBL9740225 0.82 GSK3B (0.56) GSK3BTOP2ATOP2BAADATPOLB
Hydrochloric Acid SCHEMBL29409478 0.81 KDM4E (0.67) GSK3BTOP2ATOP2BAADATPOLB
Hydrochloric Acid SCHEMBL8684414 0.81 GSK3B (0.55) GSK3BTOP2ATOP2BAADATPOLB
SCHEMBL6973262 0.81 CACNA1F (0.53) GSK3BTOP2ATOP2BPOLBCACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0924213-B1 PYRIDOBENZOXAZINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2006-06-28 EP disclosed
US-6191129-B1 MICROBIOCIDES, BACTERICIDES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2001-02-20 US disclosed
EP-0924213-A1 PYRIDOBENZOXAZINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1999-06-23 EP disclosed