SCHEMBL601078

SCHEMBL601078

Cc1c[n+]([O-])ccc1OCCCCCCCCO

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
TLR8 Q9NR97 1/20 0.34
GPR84 Q9NQS5 4/20 0.34
KDM4E B2RXH2 2/20 0.34
VDR P11473 1/20 0.33
LOX P28300 1/20 0.33
AOC3 Q16853 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
ESR1 P03372 2/20 0.33
CNR2 P34972 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL600127 0.86 GPR84 (0.36) ALDH1A1GPR84KDM4EPTGDR2CYP2D6
SCHEMBL601767 0.84 ESR1 (0.40) ALDH1A1GPR84KDM4EESR1CYP2C19
SCHEMBL600103 0.80 GPR84 (0.37) ALDH1A1GPR84KDM4EPTGDR2CA2
SCHEMBL599996 0.78 GPR84 (0.34) GPR84PTGDR2CYP2D6CYP2C19
SCHEMBL1733367 0.75 LOX (0.36) ALDH1A1TLR8KDM4ELOXAOC3
SCHEMBL1734021 0.75 LOX (0.36) ALDH1A1TLR8KDM4ELOXAOC3
SCHEMBL1735039 0.75 LOX (0.36) ALDH1A1TLR8KDM4ELOXAOC3
SCHEMBL1734201 0.75 LOX (0.36) ALDH1A1TLR8KDM4ELOXAOC3
SCHEMBL1733371 0.75 LOX (0.36) ALDH1A1TLR8KDM4ELOXAOC3
SCHEMBL1735599 0.75 LOX (0.36) ALDH1A1TLR8KDM4ELOXAOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2420500-A1 PYRIDINE THIO DERIVATIVE, AND PHARMACEUTICAL COMPOSITION WHICH CONTAINS SAME AND HAS ANTI-HELICOBACTER PYLORI ACTION aRigen Pharmaceuticals, Inc. (JP) 2012-02-22 EP disclosed
US-20120041030-A1 PYRIDINE THIO DERIVATIVE, AND PHARMACEUTICAL COMPOSITION WHICH CONTAINS SAME AND HAS ANTI-HELICOBACTER PYLORI ACTION LINK GENOMICS, INC. (JP) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120041030-A1 PYRIDINE THIO DERIVATIVE, AND PHARMACEUTICAL COMPOSITION WHICH CONTAINS SAME AND HAS ANTI-HELICOBACTER PYLORI ACTION TPMT, TST, PTPN11 ALDH1A1 1770/4885TLR8 1180/4885GPR84 3620/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.