SCHEMBL6012204

SCHEMBL6012204

CSC1=Nc2ccccc2-c2[nH]c3ccccc3c2C1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.76
CCNB2 O95067 3/20 0.76
CCNB1 P14635 3/20 0.76
GSK3B P49841 3/20 0.76
CCNB3 Q8WWL7 3/20 0.76
CA1 P00915 14/20 0.51
CA2 P00918 14/20 0.51
CA4 P22748 14/20 0.51
CA6 P23280 14/20 0.51
CCNT1 O60563 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CDK9 P50750 1/20 0.45
CCNA1 P78396 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.45
SIRT1 Q96EB6 1/20 0.45
AURKA O14965 1/20 0.42
AURKB Q96GD4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6102492 0.86 CDK1 (1.00) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL11406516 0.69 CCNB2 (0.45) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL6012236 0.69 CA1 (0.50) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL29370925 0.69 CA1 (1.00) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL2298597 0.69 CA1 (1.00) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL17963741 0.67 CA1 (0.67) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL15264467 0.65 GSK3B (0.75) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL12274879 0.65 CDK2 (0.48) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL10026452 0.65 HRH4 (0.40) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL8523044 0.64 CA1 (0.67) CDK1CCNB2CCNB1GSK3BCCNB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610684-B2 Antiproliferative agents THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2003-08-26 US claimed
EP-1086105-B1 FUSED AZEPINONE CYCLIN DEPENDENT KINASE INHIBITORS US GOV HEALTH & HUMAN SERV (US) 2006-03-01 EP disclosed