SCHEMBL6012236

SCHEMBL6012236

C1=Nc2ccccc2-c2[nH]c3ccccc3c2C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 11/20 0.50
CA2 P00918 11/20 0.50
CA4 P22748 11/20 0.50
CA6 P23280 11/20 0.50
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
TDP1 Q9NUW8 2/20 0.46
ALOX15 P16050 1/20 0.46
CDK1 P06493 3/20 0.43
CCNB2 O95067 2/20 0.43
CCNB1 P14635 2/20 0.43
GSK3B P49841 2/20 0.43
CCNB3 Q8WWL7 2/20 0.43
CDK2 P24941 2/20 0.43
CCNT1 O60563 1/20 0.43
CCNA2 P20248 1/20 0.43
CDK9 P50750 1/20 0.43
CCNA1 P78396 1/20 0.43
CDK5 Q00535 1/20 0.43
CDK5R1 Q15078 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15270863 0.84 CDK1 (0.60) CA1CA2CA4CA6MEN1
SCHEMBL7219608 0.81 GSK3B (0.54) CDK1CCNB2CCNB1GSK3BCCNB3
SCHEMBL30394416 0.73 KMT2A (0.40) CA1CA2CA4CA6KMT2A
SCHEMBL12274879 0.70 CDK2 (0.48) CA1CA2CA4CA6MEN1
SCHEMBL6012204 0.69 CDK1 (0.76) CA1CA2CA4CA6CDK1
SCHEMBL2298597 0.67 CA1 (1.00) CA1CA2CA4CA6MEN1
SCHEMBL29370925 0.67 CA1 (1.00) CA1CA2CA4CA6MEN1
SCHEMBL25235469 0.66 HTR2A (0.47) CA1CA2CA4CA6MEN1
SCHEMBL12126575 0.66 CA1 (0.71) CA1CA2CA4CA6MEN1
SCHEMBL30063877 0.66 CA1 (0.71) CA1CA2CA4CA6MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008042867-A2 MODULATORS OF MULTIPLE KINASES EMILIEM INC. (US) 2008-04-10 WO disclosed
EP-1086105-B1 FUSED AZEPINONE CYCLIN DEPENDENT KINASE INHIBITORS US GOV HEALTH & HUMAN SERV (US) 2006-03-01 EP disclosed