SCHEMBL7219608

SCHEMBL7219608

FC(F)(F)c1ccc2[nH]c3c(c2c1)CC=Nc1ccccc1-3

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 13/20 0.54
CDK5 Q00535 12/20 0.54
CDK5R1 Q15078 12/20 0.54
CDK1 P06493 12/20 0.54
CCNB2 O95067 11/20 0.54
CCNB1 P14635 11/20 0.54
CCNB3 Q8WWL7 11/20 0.54
KIF11 P52732 3/20 0.49
MDH2 P40926 1/20 0.47
GSK3A P49840 2/20 0.45
MPL P40238 1/20 0.43
CHUK O15111 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6012236 0.81 CA1 (0.50) GSK3BCDK5CDK5R1CDK1CCNB2
SCHEMBL15270863 0.81 CDK1 (0.60) GSK3BCDK5CDK5R1CDK1CCNB2
SCHEMBL5688281 0.70 GSK3B (1.00) GSK3BCDK5CDK5R1CDK1CCNB2
SCHEMBL4130017 0.67 KIF11 (1.00) KIF11CHUK
SCHEMBL27354120 0.66 KIF11 (0.56) GSK3BCDK5CDK5R1CDK1CCNB2
SCHEMBL29507666 0.65 KIF11 (0.81) KIF11CHUK
SCHEMBL412032 0.65 KIF11 (0.81) KIF11CHUK
SCHEMBL28372461 0.64 GPR3 (0.49) KIF11
SCHEMBL16085082 0.64 GSK3B (0.85) GSK3BCDK5CDK5R1CDK1CCNB2
SCHEMBL2289172 0.64 KIF11 (0.61) GSK3BCDK5CDK5R1CDK1CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6610684-B2 Antiproliferative agents THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES 2003-08-26 US claimed