SCHEMBL6012248

SCHEMBL6012248

Cc1nn(-c2ccccc2)c(C)c1CN1CCC2(CC1)C(=O)NC(Cc1ccccc1)C(=O)N2Cc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.63
CXCR3 P49682 1/20 0.57
SMO Q99835 1/20 0.44
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6012352 0.91 CCR5 (0.77) CCR5CXCR3
SCHEMBL6012398 0.91 CCR5 (0.72) CCR5
SCHEMBL6012381 0.90 CCR5 (0.62) CCR5CXCR3SMO
SCHEMBL6614696 0.88 CCR5 (0.81) CCR5
SCHEMBL6613627 0.87 CCR5 (0.66) CCR5
SCHEMBL6615034 0.86 CCR5 (0.65) CCR5
SCHEMBL6013012 0.85 CCR5 (0.63) CCR5
SCHEMBL6610385 0.84 CCR5 (0.64) CCR5
SCHEMBL6612925 0.84 CCR5 (0.62) CCR5
SCHEMBL6012745 0.83 CCR5 (0.55) CCR5CXCR3SMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119091-B2 Triazaspiro[5.5]undecane derivatives and pharmaceutical compositions comprising thereof, as an active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2006-10-10 US disclosed
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed