SCHEMBL6012352

SCHEMBL6012352

CCCCN1C(=O)C(Cc2ccccc2)NC(=O)C12CCN(Cc1c(C)nn(-c3ccccc3)c1C)CC2

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.77
CXCR3 P49682 1/20 0.60
CXCR4 P61073 2/20 0.52
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6012923 0.92 CCR5 (0.79) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012248 0.91 CCR5 (0.63) CCR5CXCR3
SCHEMBL6012381 0.90 CCR5 (0.62) CCR5CXCR3CYP3A4CYP2D6CYP2C9
SCHEMBL6613211 0.90 CCR5 (0.76) CCR5CXCR4CYP3A4CYP2D6CYP2C9
SCHEMBL5345628 0.88 CCR5 (0.76) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL5346104 0.88 CCR5 (0.77) CCR5CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6641804 0.88 CCR5 (0.77) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012919 0.88 CCR5 (0.98) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012611 0.88 CCR5 (0.98) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012520 0.88 CCR5 (0.98) CCR5CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119091-B2 Triazaspiro[5.5]undecane derivatives and pharmaceutical compositions comprising thereof, as an active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2006-10-10 US disclosed
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed