SCHEMBL6012256

SCHEMBL6012256

COCCN1C(=O)[C@H](COCC2CCCCC2)NC(=O)C12CCN(Cc1ccc(Oc3ccccc3)cc1)CC2

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.68
CYP3A4 P08684 3/20 0.68
CYP2C9 P11712 3/20 0.68
CYP2D6 P10635 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6613208 0.91 CCR5 (0.83) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6012345 0.87 CXCR3 (0.68) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6013095 0.84 CCR5 (0.85) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6012373 0.83 CCR5 (0.68) CCR5CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL5612112 0.83 CCR5 (0.85) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL2451944 0.82 CCR5 (0.98) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6012634 0.82 CCR5 (0.98) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6013122 0.81 CCR5 (0.84) CCR5CYP3A4CYP2C9CYP2D6
Hydrochloric Acid SCHEMBL5612365 0.81 CCR5 (1.00) CCR5CYP3A4CYP2C9CYP2D6
SCHEMBL6012909 0.81 CXCR3 (0.69) CCR5CYP3A4CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119091-B2 Triazaspiro[5.5]undecane derivatives and pharmaceutical compositions comprising thereof, as an active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2006-10-10 US disclosed
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed