SCHEMBL6012469

SCHEMBL6012469

C=CCOc1ccc(CN2CCC3(CC2)C(=O)NC(CC(C)C)C(=O)N3CCC)cc1

nearest known ligand 0.74

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.74
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
CYP2C9 P11712 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6610832 0.96 CCR5 (0.76) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6611577 0.87 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL2084808 0.87 CXCR3 (0.73) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6615793 0.87 CCR5 (0.75) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6611838 0.87 CCR5 (0.75) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6612347 0.86 CCR5 (0.82) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012328 0.86 CCR5 (0.81) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6012687 0.85 CCR5 (1.00) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6613169 0.85 CCR5 (0.72) CCR5CYP3A4CYP2D6CYP2C9
SCHEMBL6612415 0.84 CCR5 (0.76) CCR5CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119091-B2 Triazaspiro[5.5]undecane derivatives and pharmaceutical compositions comprising thereof, as an active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2006-10-10 US disclosed
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed