SCHEMBL6012861

SCHEMBL6012861

O=C1C(COCc2ccccc2)NC(=O)C2(CCN(CCc3ccccc3)CC2)N1CC(c1ccccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 19/20 0.51
CXCR4 P61073 2/20 0.50
OPRM1 P35372 1/20 0.47
KCNH2 Q12809 1/20 0.47
SIGMAR1 Q99720 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6012886 0.94 CCR5 (0.56) CCR5CXCR4
SCHEMBL6012554 0.94 CCR5 (0.59) CCR5CXCR4
SCHEMBL6012496 0.93 CCR5 (0.61) CCR5CXCR4
SCHEMBL6615561 0.93 CCR5 (0.61) CCR5CXCR4
SCHEMBL6616345 0.90 CCR5 (0.60) CCR5
SCHEMBL6012671 0.90 CCR5 (0.55) CCR5CXCR4OPRM1KCNH2SIGMAR1
SCHEMBL6614717 0.89 CCR5 (0.51) CCR5CXCR4
SCHEMBL6614956 0.88 CXCR3 (0.57) CCR5CXCR4
SCHEMBL6613787 0.88 CCR5 (0.59) CCR5CXCR4OPRM1KCNH2SIGMAR1
SCHEMBL6611869 0.87 CCR5 (0.58) CCR5CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119091-B2 Triazaspiro[5.5]undecane derivatives and pharmaceutical compositions comprising thereof, as an active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2006-10-10 US disclosed
EP-1236726-B1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2004-12-01 EP disclosed
EP-1236726-A1 TRIAZASPIRO 5.5]UNDECANE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-04 EP disclosed