SCHEMBL6013386

SCHEMBL6013386

CC(C)(C)c1c(N)nc(N)nc1N

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
HSD17B10 Q99714 1/20 0.35
DHFR P00374 3/20 0.33
KCNH2 Q12809 1/20 0.33
CDK1 P06493 2/20 0.32
CCNB1 P14635 2/20 0.32
CCNE1 P24864 2/20 0.32
CDK2 P24941 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21585430 0.83 L3MBTL1 (0.32) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL1774048 0.83 L3MBTL1 (0.36) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL15504760 0.74 KDM4E (0.42) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL16229312 0.72 L3MBTL1 (0.40) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL24310168 0.72 HSP90AA1 (0.39) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL3563625 0.67 HSP90AA1 (0.41) KDM4EHSD17B10DHFR
SCHEMBL28120669 0.67 HRH4 (0.50) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL20198717 0.67 HRH4 (0.50) L3MBTL1KDM4EGAAMAPTNPC1
SCHEMBL10049719 0.65 LMNA (0.39) KDM4ECDK2
SCHEMBL10635090 0.64 HSP90AA1 (0.33) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1631260-A2 PHARMACEUTICAL CO-CRYSTAL COMPOSITIONS OF DRUGS SUCH AS CARBAMAZEPINE, CELECOXIB, OLANZAPINE, ITRACONAZOLE, TOPIRAMATE, MODAFINIL, 5-FLUOROURACIL, HYDROCHLOROTHAZIDE, ACETAMINOPHEN, ASPIRIN, FLURBIPROFEN, PHENYTOIN AND IBUPROFEN Transform Pharmaceuticals, Inc. (US) 2006-03-08 EP claimed
WO-2004078163-A2 PHARMACEUTICAL CO-CRYSTAL COMPOSITIONS OF DRUGS SUCH AS CARBAMAZEPINE, CELECOXIB, OLANZAPINE, ITRACONAZOLE, TOPIRAMATE, MODAFINIL, 5-FLUOROURACIL, HYDROCHLOROTHIAZIDE, ACETAMINOPHEN, ASPIRIN, FLURBIPROFEN, PHENYTOIN AND IBUPROFEN TRANSFORM PHARMACEUTICALS, INC. (US) 2004-09-16 WO claimed