SCHEMBL6014087

SCHEMBL6014087

CCOC(=O)c1ccc(NC(=O)N(C)c2ccc(Cl)c(C(F)(F)F)c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CETP P11597 3/20 0.52
RAB9A P51151 3/20 0.51
NPC1 O15118 2/20 0.51
TP53 P04637 1/20 0.51
POLB P06746 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
SENP1 Q9P0U3 1/20 0.49
PDK1 Q15118 1/20 0.47
PDK2 Q15119 1/20 0.47
PDK3 Q15120 1/20 0.47
PDK4 Q16654 1/20 0.47
TRPV1 Q8NER1 3/20 0.46
RAF1 P04049 1/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TSHR P16473 1/20 0.46
MAPT P10636 2/20 0.46
CASP3 P42574 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
BRAF P15056 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL620123 0.82 KDR (0.67) SMN1; SMN2PDK1PDK2PDK3PDK4
SCHEMBL27823104 0.81 MLYCD (0.56) RAB9ANPC1SMN1; SMN2PDK1TRPV1
SCHEMBL16628055 0.80 RAF1 (0.63) TRPV1RAF1MEN1KMT2ABRAF
SCHEMBL10222082 0.79 KDR (0.59) PDK1TRPV1RAF1MEN1KMT2A
SCHEMBL1513766 0.78 CETP (0.44) CETPPDK2MEN1KMT2ATSHR
SCHEMBL11810258 0.78 LMNA (0.54) SMN1; SMN2KMT2ATSHRMAPTALDH1A1
SCHEMBL403261 0.78 CA12 (0.51) RAB9ATP53MAPTBRAFALDH1A1
SCHEMBL16628095 0.75 TRPV1 (0.65) PDK1TRPV1RAF1
SCHEMBL12020252 0.75 RAF1 (0.61) RAF1MEN1KMT2ABRAFHDAC1
SCHEMBL19668025 0.72 MEN1 (0.61) SMN1; SMN2RAF1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298311-B1 w-Carboxy aryl substituted diphenyl ureas as p38 kinase inhibitors BAYER HEALTHCARE LLC (US) 2012-05-09 EP disclosed