SCHEMBL6014732

SCHEMBL6014732

COc1ccc(Oc2ccc(N)cc2)cc1C(N)=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 2/20 0.53
SMN1; SMN2 Q16637 3/20 0.50
MAPT P10636 4/20 0.47
HTT P42858 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TEAD4 Q15561 1/20 0.46
ALDH1A1 P00352 6/20 0.45
TDP1 Q9NUW8 2/20 0.44
POLB P06746 2/20 0.44
MEN1 O00255 1/20 0.44
MITF O75030 1/20 0.44
GAA P10253 1/20 0.44
GFER P55789 1/20 0.44
KMT2A Q03164 1/20 0.44
NLRP1 Q9C000 1/20 0.44
NOD2 Q9HC29 1/20 0.44
CYP3A4 P08684 1/20 0.44
TSHR P16473 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HDAC3 O15379 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14538979 0.89 AR (0.49) PARP10SMN1; SMN2MAPTHTTNPSR1
SCHEMBL258010 0.84 BRAF (0.58) SMN1; SMN2MAPTHTTNPSR1ALDH1A1
SCHEMBL31295589 0.83 ALDH1A1 (0.58) MAPTHTTALDH1A1MEN1GAA
SCHEMBL623759 0.83 ALDH1A1 (0.58) MAPTHTTALDH1A1MEN1GAA
SCHEMBL1086016 0.83 MAPT (0.66) PARP10MAPTHTTNPSR1ALDH1A1
SCHEMBL30052013 0.83 MAPT (0.66) PARP10MAPTHTTNPSR1ALDH1A1
Hydrochloric Acid SCHEMBL15486584 0.82 ALDH1A1 (0.56) MAPTHTTALDH1A1TDP1POLB
Hydrochloric Acid SCHEMBL27585316 0.82 MAPT (0.64) PARP10MAPTHTTNPSR1ALDH1A1
SCHEMBL177818 0.81 SMN1; SMN2 (0.61) SMN1; SMN2MAPTTEAD4ALDH1A1TDP1
SCHEMBL31557923 0.81 PARP10 (0.56) PARP10SMN1; SMN2MAPTTEAD4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298311-B1 w-Carboxy aryl substituted diphenyl ureas as p38 kinase inhibitors BAYER HEALTHCARE LLC (US) 2012-05-09 EP disclosed