SCHEMBL6015975

SCHEMBL6015975

CN(C)CCCOC(=O)c1ccc2[c]c[nH]c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.53
ALDH1A1 P00352 3/20 0.50
PHLPP2 Q6ZVD8 1/20 0.43
MAPK1 P28482 3/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPT P10636 1/20 0.40
ESR1 P03372 1/20 0.40
LMNA P02545 3/20 0.39
SCN1A P35498 3/20 0.39
SCN2A Q99250 3/20 0.39
SCN3A Q9NY46 3/20 0.39
CYP1A2 P05177 2/20 0.39
DRD3 P35462 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KCNH2 Q12809 2/20 0.39
MAOA P21397 1/20 0.39
CNR1 P21554 1/20 0.39
DRD4 P21917 1/20 0.39
ACHE P22303 1/20 0.39
HRH2 P25021 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015765 0.93 PHLPP2 (0.51) GAAALDH1A1PHLPP2MAPK1MAPT
SCHEMBL5542394 0.86 ESR1 (0.54) ALDH1A1MAPK1MAPTESR1LMNA
SCHEMBL5539416 0.85 ESR1 (0.50) ALDH1A1MAPK1MAPTESR1LMNA
SCHEMBL5535885 0.84 ALDH1A1 (0.52) ALDH1A1MAPK1MAPTESR1LMNA
SCHEMBL5536597 0.83 ALDH1A1 (0.49) ALDH1A1MAPK1ESR1LMNACYP1A2
SCHEMBL5540470 0.80 CA12 (0.50) ALDH1A1MAPK1HSD17B10MAPTESR1
SCHEMBL6015708 0.78 KDM4E (0.55) ALDH1A1HSD17B10KDM4ERAB9AKMT2A
SCHEMBL9629064 0.77 GAA (0.84) GAAALDH1A1PHLPP2MAPK1HSD17B10
SCHEMBL6015768 0.77 KDM4E (0.47) ALDH1A1MAOAHRH3HTR1AKDM4E
SCHEMBL27601533 0.76 ESR1 (0.38) ALDH1A1MAPK1HSD17B10MAPTESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN disclosed