SCHEMBL6016367

SCHEMBL6016367

COc1cc(CN(C)C(=O)c2cnc(OCCN(C)C)nc2-c2ccccc2C)cc(OC)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 7/20 0.47
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
PIK3CD O00329 1/20 0.37
ROCK2 O75116 3/20 0.37
ROCK1 Q13464 3/20 0.37
WDR5 P61964 2/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016394 0.80 KDM4E (0.43)
SCHEMBL6016339 0.78 CHRM2 (0.43) KMT2A
Dimethylaminoethanol SCHEMBL6016335 0.76 ALDH1A1 (0.43)
SCHEMBL6016503 0.74 KDM4E (0.41)
SCHEMBL6016603 0.73 TACR1 (0.50) TACR1
SCHEMBL7704059 0.70 TACR1 (0.51) TACR1HSP90AA1HSP90AB1KMT2A
SCHEMBL6016671 0.69 TACR1 (0.49) TACR1
SCHEMBL6016572 0.69 MAPK14 (0.48) KMT2A
SCHEMBL6866620 0.68 ALDH1A1 (0.44)
SCHEMBL6016508 0.68 KDM4E (0.38) HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed