SCHEMBL6016502

SCHEMBL6016502

CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)Oc1cnc(N2CCOCC2)nc1-c1ccccc1Br

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 15/20 0.53
RAF1 P04049 3/20 0.41
BRAF P15056 3/20 0.41
AOC3 Q16853 1/20 0.40
CETP P11597 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016428 0.91 TACR1 (0.64) TACR1
SCHEMBL6016461 0.91 TACR1 (0.64) TACR1RAF1BRAF
SCHEMBL6016612 0.91 TACR1 (0.54) TACR1RAF1BRAFAOC3CETP
SCHEMBL6016498 0.91 TACR1 (0.53) TACR1
SCHEMBL6016479 0.91 TACR1 (0.53) TACR1RAF1BRAFAOC3CETP
SCHEMBL6016561 0.90 TACR1 (0.52) TACR1RAF1BRAFAOC3CETP
SCHEMBL6016505 0.86 TACR1 (0.48) TACR1CETP
SCHEMBL6016548 0.85 TACR1 (0.54) TACR1RAF1BRAF
SCHEMBL6016733 0.83 TACR1 (0.65) TACR1
SCHEMBL6016699 0.83 TACR1 (0.65) TACR1BRAFCETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP claimed