SCHEMBL6016548

SCHEMBL6016548

Cc1cc(F)ccc1-c1nc(N2CCOCC2)ncc1OC(=O)N(C)Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 12/20 0.54
RAF1 P04049 8/20 0.44
BRAF P15056 8/20 0.44
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016610 0.91 TACR1 (0.54) TACR1CYP3A4CYP2D6CYP2C9
SCHEMBL6016461 0.91 TACR1 (0.64) TACR1RAF1BRAF
SCHEMBL6016612 0.88 TACR1 (0.54) TACR1RAF1BRAF
SCHEMBL6016693 0.86 TACR1 (0.49) TACR1CYP3A4CYP2D6CYP2C9
SCHEMBL6016502 0.85 TACR1 (0.53) TACR1RAF1BRAF
SCHEMBL6016479 0.85 TACR1 (0.53) TACR1RAF1BRAF
SCHEMBL6016561 0.85 TACR1 (0.52) TACR1RAF1BRAF
SCHEMBL6016649 0.82 TACR1 (0.77) TACR1BRAF
SCHEMBL6016476 0.81 TACR1 (0.64) TACR1
SCHEMBL6016547 0.81 TACR1 (0.57) TACR1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP claimed