SCHEMBL6016479

SCHEMBL6016479

CN(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)C(=O)Oc1cnc(N2CCOCC2)nc1-c1ccccc1Cl

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.53
CETP P11597 2/20 0.44
RAF1 P04049 3/20 0.41
BRAF P15056 3/20 0.41
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
AOC3 Q16853 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016612 0.91 TACR1 (0.54) TACR1CETPRAF1BRAFTDP1
SCHEMBL6016461 0.91 TACR1 (0.64) TACR1RAF1BRAF
SCHEMBL6016586 0.91 TACR1 (0.64) TACR1
SCHEMBL6016502 0.91 TACR1 (0.53) TACR1CETPRAF1BRAFAOC3
SCHEMBL6016604 0.91 TACR1 (0.53) TACR1
SCHEMBL6016561 0.90 TACR1 (0.52) TACR1CETPRAF1BRAFAOC3
SCHEMBL6016483 0.86 TACR1 (0.48) TACR1
SCHEMBL6016582 0.86 TACR1 (0.44) TACR1RAF1BRAF
SCHEMBL6016548 0.85 TACR1 (0.54) TACR1RAF1BRAF
SCHEMBL6016699 0.83 TACR1 (0.65) TACR1CETPBRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP claimed