SCHEMBL6017148

SCHEMBL6017148

Cc1nc(-c2ccc(C(F)(F)F)cc2)ccc1CCOc1ccc2[nH]cc(CC(=O)OC(C)(C)C)c2c1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.44
MTNR1A P48039 7/20 0.43
MTNR1B P49286 6/20 0.43
PPARA Q07869 4/20 0.40
PPARG P37231 3/20 0.40
PPARD Q03181 2/20 0.40
ICMT O60725 1/20 0.39
KDM4E B2RXH2 1/20 0.39
LTA4H P09960 2/20 0.38
PLA2G2A P14555 2/20 0.38
HCRTR2 O43614 1/20 0.38
NR1H2 P55055 1/20 0.38
NR1H3 Q13133 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5617384 0.84 PPARD (0.45) TRPV1PPARAPPARGPPARDKDM4E
SCHEMBL5669972 0.79 PPARD (0.41) PPARAPPARGPPARDNR1H2NR1H3
SCHEMBL6052634 0.78 PPARD (0.52) PPARAPPARGPPARD
SCHEMBL6029170 0.77 MCL1 (0.41) PPARAPPARGPPARD
SCHEMBL6030489 0.77 PPARD (0.48) PPARAPPARGPPARD
SCHEMBL6052594 0.77 PPARA (0.44) PPARAPPARGPPARD
SCHEMBL5617387 0.77 PPARD (0.49) PPARAPPARGPPARDNR1H2NR1H3
SCHEMBL6017372 0.76 PKM (0.43) TRPV1PPARAPPARGPPARD
SCHEMBL6052586 0.76 PPARD (0.51) PPARAPPARGPPARD
SCHEMBL6218546 0.76 PPARD (0.59) PPARAPPARGPPARDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed