SCHEMBL6017372

SCHEMBL6017372

CCOC(=O)Cc1c[nH]c2cc(OCc3ccc(-c4ccc(C(F)(F)F)cc4)nc3C)ccc12

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.43
PPARD Q03181 10/20 0.42
PPARA Q07869 6/20 0.42
PPARG P37231 2/20 0.39
MAOB P27338 2/20 0.39
IGF1R P08069 1/20 0.37
MET P08581 1/20 0.37
SRC P12931 1/20 0.37
ESR1 P03372 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
PRMT5 O14744 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017323 0.93 PKM (0.45) PKMPPARDPPARAMAOBIGF1R
SCHEMBL5617387 0.91 PPARD (0.49) PPARDPPARAPPARG
SCHEMBL6017227 0.88 PKM (0.41) PKMPPARDPPARAPPARGMAOB
SCHEMBL6017361 0.86 PKM (0.42) PKMPPARDPPARAPPARGMAOB
SCHEMBL6017265 0.85 PKM (0.42) PKMPPARDTRPV1PRMT5
SCHEMBL6064609 0.84 PKM (0.42) PKMPPARDPPARAPPARGMAOB
SCHEMBL5617384 0.83 PPARD (0.45) PPARDPPARAPPARGTRPV1
SCHEMBL6065369 0.82 PKM (0.40) PKMPPARDPPARAPPARGMAOB
SCHEMBL6017371 0.81 TRPV1 (0.45) PKMPPARDPPARAPPARGMAOB
SCHEMBL6017580 0.80 MAOB (0.40) PKMPPARDPPARAMAOBIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed