SCHEMBL6017301

SCHEMBL6017301

F[CH]Cc1ccc(Br)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.44
TAAR1 Q96RJ0 3/20 0.44
HTR2A P28223 1/20 0.44
IDO1 P14902 4/20 0.42
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
PYCR1 P32322 3/20 0.38
PLCG1 P19174 1/20 0.37
TGM2 P21980 1/20 0.36
MAOB P27338 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13673478 0.78 CYP2A6 (0.44) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL20103 0.78 CYP2A6 (0.44) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL648420 0.76 ALDH1A1 (0.52) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL28879807 0.76 TAAR1 (0.42) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL11306664 0.76 ESR1 (0.50) TAAR1IDO1MEN1KMT2A
SCHEMBL219760 0.74
SCHEMBL28743524 0.74 IDO1 (0.44) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL24042960 0.72 IDO1 (0.43) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL3255735 0.72 IDO1 (0.43) CYP2A6TAAR1HTR2AIDO1MEN1
SCHEMBL9680305 0.72 ALDH1A1 (0.44) CYP2A6TAAR1HTR2AIDO1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551834-A4 SUBSTITUTED QUINAZOLINONE COMPOUNDS CHIRON CORP (US) 2006-08-23 EP disclosed
EP-1551834-A1 SUBSTITUTED QUINAZOLINONE COMPOUNDS CHIRON CORPORATION (US) 2005-07-13 EP disclosed
WO-2003099818-A1 SUBSTITUTED QUINAZOLINONE COMPOUNDS CHIRON CORPORATION (US) 2003-12-04 WO disclosed