SCHEMBL6017332

SCHEMBL6017332

Cc1nc(-c2ccc(C(F)(F)F)cc2)ncc1CN(C)c1ccc2[nH]cc(CC(=O)O)c2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ICMT O60725 2/20 0.41
TSHR P16473 2/20 0.40
LMNA P02545 3/20 0.39
ALDH1A1 P00352 2/20 0.39
GLA P06280 2/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
NFKB1 P19838 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PPARD Q03181 5/20 0.38
PIM1 P11309 4/20 0.37
PIM3 Q86V86 4/20 0.37
NR1H2 P55055 1/20 0.37
NR1H3 Q13133 1/20 0.37
PPARA Q07869 4/20 0.37
PPARG P37231 2/20 0.37
SNCA P37840 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017109 0.91 TRPV1 (0.42) ICMTLMNAALDH1A1GLACYP2C9
SCHEMBL5617133 0.83 KDM4E (0.48) ICMTTSHRLMNAALDH1A1GLA
SCHEMBL5630993 0.76 PPARD (0.48) PPARDPPARAPPARG
SCHEMBL6017371 0.74 TRPV1 (0.45) ICMTLMNATRPV1PPARDPPARA
SCHEMBL6017333 0.73 TRPV1 (0.48) ICMTTRPV1KDM4EPPARDPPARA
SCHEMBL6017240 0.72 KDM4E (0.43) ICMTTSHRLMNAALDH1A1GLA
SCHEMBL6017456 0.71 GRIN2B (0.43) NFKB1PPARDPPARAPPARG
SCHEMBL27642697 0.71 GRIN1 (0.40) NFKB1PPARDPPARAPPARG
SCHEMBL6287980 0.71 TSHR (0.67) ICMTTSHRLMNAALDH1A1GLA
SCHEMBL6489229 0.69 PPARD (0.70) PPARDPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed