SCHEMBL6017240

SCHEMBL6017240

O=C(O)Cc1c[nH]c2ccc(OCc3cnc(-c4ccc(C(F)(F)F)cc4)nc3C3CC3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
PPARD Q03181 12/20 0.42
PPARA Q07869 8/20 0.42
PPARG P37231 2/20 0.42
TRPV1 Q8NER1 1/20 0.41
ICMT O60725 1/20 0.40
TSHR P16473 2/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
GLA P06280 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
NFKB1 P19838 1/20 0.39
PMP22 Q01453 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MEN1 O00255 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
LTA4H P09960 1/20 0.38
PLA2G2A P14555 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5617383 0.94 PPARD (0.43) PPARDPPARAPPARG
SCHEMBL6017387 0.90 TRPV1 (0.40) KDM4EPPARDPPARAPPARGTRPV1
SCHEMBL5617133 0.87 KDM4E (0.48) KDM4EPPARDPPARAPPARGTRPV1
SCHEMBL6017141 0.86 PPARA (0.39) PPARDPPARAPPARGTRPV1
SCHEMBL6017580 0.84 MAOB (0.40) PPARDPPARATRPV1NFKB1
SCHEMBL6017333 0.83 TRPV1 (0.48) KDM4EPPARDPPARAPPARGTRPV1
SCHEMBL1227421 0.80 PTGDR2 (0.41)
SCHEMBL6017371 0.78 TRPV1 (0.45) PPARDPPARAPPARGTRPV1ICMT
SCHEMBL1549165 0.78 PPARD (0.59) PPARDPPARAPPARG
SCHEMBL6017772 0.77 PPARD (0.55) PPARDPPARAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed