SCHEMBL6017759

SCHEMBL6017759

CCN(CC)CCCC(C)Nc1ccc(S(=O)(=O)Oc2ccc3[nH]c(N(C=O)C4CC4)nc3c2)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.35
CCR4 P51679 4/20 0.35
TMEM97 Q5BJF2 1/20 0.35
SIGMAR1 Q99720 1/20 0.35
KCNH3 Q9ULD8 1/20 0.34
MELK Q14680 1/20 0.34
USP2 O75604 4/20 0.33
TP53 P04637 3/20 0.33
CYP3A4 P08684 3/20 0.33
CASP1 P29466 3/20 0.33
CASP7 P55210 3/20 0.33
HBB P68871 3/20 0.33
HSD17B10 Q99714 3/20 0.33
APP P05067 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
BRCA1 P38398 2/20 0.33
HIF1A Q16665 2/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017614 0.86 EGFR (0.32)
SCHEMBL6018066 0.82 ENPP3 (0.31) KDM4EALDH1A1
SCHEMBL5041061 0.81 ENPP3 (0.39) USP2TP53CYP3A4CASP1CASP7
SCHEMBL7044189 0.78 ENPP3 (0.33) KDM4EALDH1A1MAPTHTT
SCHEMBL6017897 0.78 ENPP3 (0.33) KDM4EMEN1KMT2AALDH1A1MAPT
SCHEMBL6018120 0.78 ENPP3 (0.30)
SCHEMBL5036606 0.77 ENPP3 (0.33) KDM4ELMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL6017698 0.76 ACE2 (0.31) TDP1MAPK1
SCHEMBL6017766 0.76 ENPP3 (0.31)
SCHEMBL6017660 0.76 ENPP3 (0.33) KDM4EMEN1KMT2AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7041668-B2 Substituted benzimidazole compounds and their use for the treatment of cancer AVENTIS PHARMA S.A. (FR) 2006-05-09 US disclosed
US-20050014811-A1 Substituted benzimidazole compounds and their use for the treatment of cancer AVENTIS PHARMA S.A. (FR) 2005-01-20 US disclosed
EP-1432417-A2 SUBSTITUTED BENZIMIDAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCER Aventis Pharma S.A. (FR) 2004-06-30 EP disclosed
WO-2003028721-A2 SUBSTITUTED BENZIMIDAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCER AVENTIS PHARMA S.A. (FR) 2003-04-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050014811-A1 Substituted benzimidazole compounds and their use for the treatment of cancer CDKL3, CCNL2, CDKL1 CXCR4 2293/4885CCR4 1501/4885TMEM97 1091/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.