SCHEMBL6018154

SCHEMBL6018154

CNC(=O)[CH]c1cccc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 2/20 0.56
HDAC8 Q9BY41 2/20 0.54
HDAC6 Q9UBN7 1/20 0.54
MTNR1A P48039 2/20 0.53
MTNR1B P49286 1/20 0.53
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
PGR P06401 1/20 0.47
GAA P10253 1/20 0.47
PTGS1 P23219 1/20 0.47
HSD17B10 Q99714 1/20 0.47
F2 P00734 1/20 0.47
LMNA P02545 1/20 0.47
MMP3 P08254 1/20 0.44
KDM4E B2RXH2 1/20 0.44
NR4A1 P22736 1/20 0.44
NR4A2 P43354 1/20 0.44
NR4A3 Q92570 1/20 0.44
NPC1 O15118 3/20 0.42
MEN1 O00255 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3245346 0.79 MTNR1A (0.57) PLK1HDAC8HDAC6MTNR1AMTNR1B
SCHEMBL5459262 0.79 MTNR1A (0.53) PLK1HDAC8HDAC6MTNR1AMTNR1B
SCHEMBL28312715 0.78 MTNR1A (0.56) PLK1HDAC8HDAC6MTNR1AMTNR1B
SCHEMBL11101904 0.77 MTNR1A (0.51) PLK1HDAC8HDAC6MTNR1AMTNR1B
SCHEMBL1086540 0.77 GRIN2D (0.53) PLK1HDAC8HDAC6MTNR1AMTNR1B
SCHEMBL5651919 0.77 NR4A1 (0.55) HDAC8HDAC6MTNR1AMTNR1BALDH1A1
SCHEMBL9059821 0.75 EGFR (0.52) ALDH1A1MAPK1HPGD
Dimethylamine SCHEMBL5859542 0.73 MTNR1A (0.50) PLK1HDAC8HDAC6MTNR1AMTNR1B
SCHEMBL3245844 0.73 CYP1A2 (0.54) HDAC8HDAC6MTNR1AMTNR1BALDH1A1
SCHEMBL10684505 0.72 HDAC8 (0.48) PLK1HDAC8HDAC6MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7098215-B2 Nitrogenous compounds and antiviral drugs containing the same KUREHA CHEMICAL INDUSTRY CO., LTD. (JP) 2006-08-29 US disclosed
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound KUREHA CORPORATION (JP) 2004-08-12 US disclosed
US-20040092556-A1 Nitrogenous compounds and antiviral drugs containing the same KUREHA CORPORATION (JP) 2004-05-13 US disclosed
EP-1389460-A1 CXCR4-ANTAGONISTIC DRUGS COMPRISING NITROGEN-CONTAINING COMPOUND Kureha Chemical Industry Co., Ltd. (JP) 2004-02-18 EP disclosed
EP-1273571-A1 NITROGENOUS COMPOUNDS AND ANTIVIRAL DRUGS CONTAINING THE SAME Kureha Chemical Industry Co., Ltd. (JP) 2003-01-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092556-A1 Nitrogenous compounds and antiviral drugs containing the same NSUN2, ZC3HAV1L, PNP PLK1 4168/4885HDAC8 2580/4885HDAC6 3064/4885
US-20040157818-A1 Cxcr4-antagonistic drugs composed of nitrogen-containing compound CXCR4, CXCR1, CXCR2 PLK1 3109/4885HDAC8 2864/4885HDAC6 1799/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.