SCHEMBL6019495

SCHEMBL6019495

Cn1c(C(F)(F)F)nc2c(Br)cccc21

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
GLA P06280 1/20 0.40
GRM2 Q14416 8/20 0.40
ENPP3 O14638 1/20 0.39
ENPP1 P22413 1/20 0.39
HSD11B1 P28845 1/20 0.38
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
MAPK1 P28482 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
BACE1 P56817 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17378584 0.81 CYP1A2 (0.40) CYP1A2GLAGRM2HSD11B1NR1H2
SCHEMBL28331893 0.80 CYP1A2 (0.40) CYP1A2GLAHSD11B1NR1H2NR1H3
SCHEMBL15000593 0.80 TLR8 (0.43) CYP1A2GLANR1H2NR1H3MAPK1
SCHEMBL15520213 0.78 CYP1A2 (0.48) CYP1A2GLAENPP3ENPP1HSD11B1
SCHEMBL6950074 0.78 TLR8 (0.44) CYP1A2GLAGRM2NPC1RAB9A
SCHEMBL7876217 0.75 SMN1; SMN2 (0.50) GRM2ENPP3ENPP1HSD11B1NPC1
SCHEMBL22286053 0.74 LMNA (0.40) CYP1A2GRM2ENPP3ENPP1ALDH1A1
SCHEMBL7887559 0.74 GRM2 (0.38) GRM2NPC1RAB9AALDH1A1MEN1
SCHEMBL31005200 0.74 MMP12 (0.47) GRM2BACE1
SCHEMBL18341299 0.74 MMP12 (0.47) GRM2BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613626-A1 CYCLIC BENZIMIDAZOLES ALTANA Pharma AG (DE) 2006-01-11 EP disclosed
WO-2004087701-A1 CYCLIC BENZIMIDAZOLES ALTANA PHARMA AG (DE) 2004-10-14 WO disclosed