SCHEMBL6023488

SCHEMBL6023488

N#Cc1cccc(-c2cc(N3CCC(CNC(=O)O)C3)nc(N)n2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.45
ADORA1 P30542 2/20 0.45
PDE4D Q08499 4/20 0.43
HRH4 Q9H3N8 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
USP30 Q70CQ3 5/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
ADRA2C P18825 1/20 0.42
HTR1D P28221 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
HTR7 P34969 1/20 0.42
AURKA O14965 2/20 0.41
PDPK1 O15530 2/20 0.41
ROCK1 Q13464 2/20 0.41
AURKB Q96GD4 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6023051 0.88 USP2 (0.52) HRH4USP30AURKAPDPK1ROCK1
SCHEMBL6510066 0.80 LMNA (0.53) ADORA2AADORA1HRH4AURKAPDPK1
SCHEMBL6023493 0.79 JAK2 (0.45) ADORA2APDE4DHRH4HRH3USP30
Hydrochloric Acid SCHEMBL604938 0.78 HRH4 (0.55) HRH4HRH3
SCHEMBL6023878 0.75 LMNA (0.55) HRH4HRH3LMNATSHRHTT
SCHEMBL5076737 0.75 LMNA (0.55) HRH4HRH3LMNATSHRHTT
SCHEMBL1775505 0.75 LMNA (0.55) HRH4HRH3LMNATSHRHTT
SCHEMBL4392707 0.75 HRH4 (0.64) HRH4HRH3
SCHEMBL12483311 0.75 CCNC (0.43) ADORA2AADORA1USP30HTR2A
SCHEMBL17745899 0.75 CCNC (0.43) ADORA2AADORA1USP30HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654237-A1 2-AMINOPYRIMIDINE DERIVATIVES Bayer HealthCare AG (DE) 2006-05-10 EP disclosed
WO-2005014556-A1 2-AMINOPYRIMIDINE DERIVATIVES BAYER HEALTHCARE AG (DE) 2005-02-17 WO disclosed
EP-1505064-A1 2-Aminopyrimidine derivatives Bayer HealthCare AG (DE) 2005-02-09 EP disclosed