SCHEMBL6024664

SCHEMBL6024664

CCCCN(N)C(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA1 P00915 5/20 0.38
CA12 O43570 4/20 0.38
CA14 Q9ULX7 3/20 0.38
HDAC6 Q9UBN7 2/20 0.38
CA7 P43166 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
CTSK P43235 5/20 0.36
CA9 Q16790 2/20 0.35
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP3 P08254 1/20 0.33
MMP8 P22894 1/20 0.33
CA2 P00918 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
CTSS P25774 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1884648 0.94 CA14 (0.40) CA1CA12CA14HDAC6CA7
SCHEMBL27947608 0.93 HDAC1 (0.39) CA1CA12CA14HDAC6CA7
SCHEMBL27868897 0.93 HDAC1 (0.39) CA1CA12CA14HDAC6CA7
SCHEMBL27662317 0.93 HDAC1 (0.39) CA1CA12CA14HDAC6CA7
SCHEMBL28085982 0.93 HDAC1 (0.39) CA1CA12CA14HDAC6CA7
SCHEMBL1512279 0.88 CA14 (0.43) CA1CA12CA14HDAC6CA7
SCHEMBL8310669 0.85 CA14 (0.41) CA1CA12CA14HDAC6CA7
SCHEMBL27942277 0.83 HDAC6 (0.37) CA1CA12CA14HDAC6CA7
SCHEMBL27910088 0.81 TDP1 (0.46) CA14HDAC6HDAC1HDAC2L3MBTL1
SCHEMBL5287476 0.81 HDAC6 (0.39) CA14HDAC6HDAC1HDAC2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116723839-A Tricyclic heterobifunctional compounds for degrading target proteins C4医药公司 2023-09-08 CN disclosed
US-20230039917-A1 EXO-AZA SPIRO INHIBITORS OF MENIN-MLL INTERACTION JANSSEN PHARMACEUTICA NV (BE) 2023-02-09 US disclosed
EP-3694836-B1 PROCESS FOR PREPARING INTERMEDIATE OF ANTI-TUMOR DRUG NIRAPARIB AND INTERMEDIATE THEREOF ZAI LAB SHANGHAI CO LTD (CN) 2022-06-15 EP disclosed
WO-2019072237-A1 PROCESS FOR PREPARING INTERMEDIATE OF ANTI-TUMOR DRUG NIRAPARIB AND INTERMEDIATE THEREOF ZAI LAB (SHANGHAI) CO., LTD. (CN) 2019-04-18 WO disclosed
CN-103717589-B For treating or prevent the compound of respiratory syncytial virus disease 弗·哈夫曼-拉罗切有限公司 2016-08-17 CN disclosed
EP-1363873-B1 PEPTIDE DEFORMYLASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2016-04-20 EP disclosed
CN-102766142-A Lactam compounds useful as protein kinase inhibitors MILLENIUM PHARMACEUTICALS INC 2012-11-07 CN disclosed
CN-101068815-B Lactam compounds useful as protein kinase inhibitors MILLENNIUM PHARM INC 2012-09-05 CN disclosed
CN-102656174-A Compounds for the treatment of hepatitis C BRISTOL MYERS SQUIBB CO 2012-09-05 CN disclosed
CN-102015717-A Chemokine receptor modulators ALTIRIS THERAPEUTICS 2011-04-13 CN disclosed
CN-1617859-A 5-sulfanyl-4H-1, 2, 4-triazole derivatives and their use as medicaments SOD CONSEILS RECH APPLIC (FR) 2005-05-18 CN disclosed
CN-1599739-A Sulfonamido substituted imidazopyridines 3M INNOVATIVE PROPERTIES CO (US) 2005-03-23 CN disclosed
CN-1599740-A Amide substituted imidazopyridines 3M INNOVATIVE PROPERTIES CO (US) 2005-03-23 CN disclosed
CN-1599738-A Urea substituted imidazopyridines 3M INNOVATIVE PROPERTIES CO (US) 2005-03-23 CN disclosed
US-20040087585-A1 Peptide deformylase inhibitors GLAXOSMITHKLINE LLC 2004-05-06 US disclosed
CN-1478090-A Substituted imidazopyridines 3M 2004-02-25 CN disclosed
EP-1363873-A2 PEPTIDE DEFORMYLASE INHIBITORS SmithKline Beecham Corporation (US) 2003-11-26 EP disclosed
WO-2002070541-A2 PEPTIDE DEFORMYLASE INHIBITORS SMITH KLINE BEECHAM CORPORATION (US) 2002-09-12 WO disclosed
CN-1306442-A Improement in or relating to contrast agents NYCOMED INAGING AS (NO) 2001-08-01 CN disclosed
CN-1039016-A N '-replacement-N, N '-two replaces the hydrazine insect repellent ROHM & HAAS (US) 1990-01-24 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040087585-A1 Peptide deformylase inhibitors PDF, DPEP1, PEPD CA1 4855/4885CA12 4861/4885CA14 4831/4885
US-20230039917-A1 EXO-AZA SPIRO INHIBITORS OF MENIN-MLL INTERACTION BMI1, MLLT1, SUZ12 CA1 4703/4885CA12 4782/4885CA14 4773/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.