SCHEMBL6028217

SCHEMBL6028217

COc1ccccc1Cc1ccc2c(c1)C(c1cccc(C(N)=O)c1)=NCC(=O)N2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.49
CHEK2 O96017 1/20 0.47
KMT2A Q03164 1/20 0.45
PDE4D Q08499 2/20 0.43
CNR1 P21554 1/20 0.43
NTSR1 P30989 1/20 0.43
OPRK1 P41145 1/20 0.43
GABRA1 P14867 3/20 0.43
GABRA5 P31644 3/20 0.43
GABRA3 P34903 3/20 0.43
GABRA2 P47869 3/20 0.43
GABRB2 P47870 3/20 0.43
GABRG2 P18507 2/20 0.43
GABRB3 P28472 2/20 0.43
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41
TUBA1B P68363 2/20 0.41
TUBA4A P68366 2/20 0.41
TUBB4B P68371 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6029083 0.91 TUBB4A (0.48) PDE2ACHEK2KMT2APDE4DCNR1
SCHEMBL4708595 0.83 PDE2A (0.55) PDE2AKMT2APDE4DCNR1NTSR1
SCHEMBL5044563 0.82 PDE2A (0.57) PDE2AKMT2APDE4DCNR1NTSR1
SCHEMBL5034754 0.79 PDE2A (0.60) PDE2ACHEK2KMT2APDE4DCNR1
SCHEMBL6028359 0.78 PDE2A (0.51) PDE2ACHEK2KMT2APDE4DCNR1
SCHEMBL6028000 0.75 PDE2A (0.46) PDE2AKMT2APDE4DCNR1NTSR1
SCHEMBL4707743 0.75 PDE2A (0.48) PDE2AKMT2APDE4DTUBB4ATUBB
SCHEMBL6028943 0.74 PDE2A (0.44) PDE2AKMT2APDE4DCNR1NTSR1
SCHEMBL5972459 0.72 TUBB4A (0.47) PDE2AKMT2APDE4DCNR1NTSR1
SCHEMBL6028512 0.71 GABRA1 (0.45) KMT2APDE4DCNR1NTSR1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697332-A1 BENZO'1,4 ! DIAZEPIN-2-ONE DERIVATIVES AS PHOSPHODIESTERASE PDE2 INHIBITORS, PREPARATION AND THERAPEUTIC USE THEREOF NEURO3D (FR) 2006-09-06 EP claimed
WO-2005063723-A1 BENZO`1,4 ! DIAZEPIN-2-ONE DERIVATIVES AS PHOSPHODIESTERASE PDE2 INHIBITORS, PREPARATION AND THERAPEUTIC USE THEREOF NEURO3D (FR) 2005-07-14 WO claimed