SCHEMBL6028503

SCHEMBL6028503

Nc1cc(N2CCCC2=O)ccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPOX P50336 1/20 0.55
SLC6A2 P23975 4/20 0.50
SLC6A4 P31645 4/20 0.50
ALDH1A1 P00352 4/20 0.50
SLC6A3 Q01959 2/20 0.50
HPGD P15428 2/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
AKR1C3 P42330 1/20 0.48
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 1/20 0.46
LMNA P02545 1/20 0.44
HSD17B10 Q99714 1/20 0.44
GAA P10253 1/20 0.43
MEN1 O00255 1/20 0.43
ATM Q13315 1/20 0.43
PRKAB2 O43741 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL12493709 0.92 PPOX (0.55) PPOXSLC6A2SLC6A4ALDH1A1SLC6A3
SCHEMBL78346 0.87 SLC6A2 (0.50) SLC6A2SLC6A4ALDH1A1SLC6A3HPGD
SCHEMBL6431344 0.86 SLC6A2 (0.65) SLC6A2SLC6A4ALDH1A1SLC6A3HPGD
SCHEMBL15157023 0.84 ALDH1A1 (0.54) ALDH1A1HPGDCYP1A2CYP3A4CYP2D6
SCHEMBL7806569 0.82 SLC6A2 (0.49) SLC6A2SLC6A4ALDH1A1SLC6A3HPGD
SCHEMBL12362768 0.82 ALDH1A1 (0.53) SLC6A2SLC6A4ALDH1A1SLC6A3HPGD
SCHEMBL7814371 0.82 ALDH1A1 (0.58) SLC6A2SLC6A4ALDH1A1SLC6A3HPGD
SCHEMBL6523537 0.80 ALDH1A1 (0.50) ALDH1A1HPGDCYP1A2CYP3A4CYP2D6
SCHEMBL6029717 0.80 ALDH1A1 (0.50) ALDH1A1HPGDCYP1A2CYP3A4CYP2D6
SCHEMBL6028329 0.80 HSD17B10 (0.59) ALDH1A1HPGDCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1723129-A1 1-AKAN-2-OL SUBSTITUTED PIPERAZINE AND PIPERIDINE COMPOUNDS CV THERAPEUTICS, INC. (US) 2006-11-22 EP disclosed
WO-2005061470-A1 1-AKAN-2-OL SUBSTITUTED PIPERAZINE AND PIPERIDINE COMPOUNDS CV THERAPEUTICS, INC. (US) 2005-07-07 WO disclosed
US-4297440-A CONTAINING A 3-ANILINO-5-PYRAZOLONE MAGENTA COUPLER FUJI PHOTO FILM CO., LTD. (JP) 1981-10-27 US disclosed