SCHEMBL6032072

SCHEMBL6032072

O=C(CCl)c1cc2ccccc2o1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 1/20 0.65
ALDH1A1 P00352 6/20 0.57
MAPT P10636 5/20 0.57
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
L3MBTL1 Q9Y468 2/20 0.57
TSHR P16473 2/20 0.57
MAPK1 P28482 2/20 0.57
MEN1 O00255 1/20 0.57
KMT2A Q03164 1/20 0.57
HTT P42858 2/20 0.55
KDM4E B2RXH2 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
HPGD P15428 4/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
TP53 P04637 3/20 0.54
PKM P14618 1/20 0.53
NFKB1 P19838 1/20 0.53
NFKB2 Q00653 1/20 0.53
RELA Q04206 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8910943 0.86 FLT3 (0.61) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL10313745 0.84 FLT3 (0.67) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL28117952 0.84 FLT3 (0.67) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL10155752 0.84 FLT3 (0.67) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL243970 0.82 FLT3 (0.65) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL14432867 0.82 FLT3 (0.65) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL7914651 0.81 FLT3 (0.59) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL2560643 0.81 FLT3 (0.62) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL5158485 0.81 FLT3 (0.62) FLT3ALDH1A1MAPTNPC1RAB9A
SCHEMBL557778 0.79 FLT3 (0.71) FLT3ALDH1A1MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060094710-A1 Piperidine-pyridazones and phthalazones as pde4 inhibitors ALTANA PHARMA AG (DE) 2006-05-04 US disclosed
EP-1556049-A1 PIPERIDINE-PYRIDAZONES AND PHTHALAZONES AS PDE4 INHIBITORS ALTANA Pharma AG (DE) 2005-07-27 EP disclosed
EP-1458719-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2004-09-22 EP disclosed
WO-2004017974-A1 PIPERIDINE-PYRIDAZONES AND PHTHALAZONES AS PDE4 INHIBITORS ALTANA PHARMA AG (DE) 2004-03-04 WO disclosed
US-20030207877-A1 Pyridoquinoxaline antivirals PHARMACIA & UPJOHN COMPANY 2003-11-06 US disclosed
WO-2003053971-A1 PYRIDOQUINOXALINE ANTIVIRALS PHARMACIA & UPJOHN COMPANY (US) 2003-07-03 WO disclosed
EP-0564924-B1 2-Oxoethyl derivatives as immunosuppressants BAYER AG (US) 1998-09-09 EP disclosed
US-5686424-A FOR TREATING INFLAMMATION MILES INC. (US) 1997-11-11 US disclosed
US-5679678-A ANALGESIC AND ANTIINFLAMMATORY AGENTS CHEMISCH PHARMAZEUTISCHE FORSCHUNGSGESELLSCHAFT M.B.H. (AT) 1997-10-21 US disclosed
EP-0658559-A1 Thienothiazin derivatives, process for their preparation and their use as 5-dipoxygenase and cyclooxygenase inhibitors Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. (AT) 1995-06-21 EP disclosed
EP-0564924-A2 2-Oxoethyl derivatives as immunosuppressants Bayer Corporation (US) 1993-10-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030207877-A1 Pyridoquinoxaline antivirals IFNAR1, SARS1, ZC3HAV1 FLT3 2159/4885ALDH1A1 1275/4885MAPT 4375/4885
US-20060094710-A1 Piperidine-pyridazones and phthalazones as pde4 inhibitors PDE4A, PDE4B, PDE3A FLT3 3927/4885ALDH1A1 88/4885MAPT 2544/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.