SCHEMBL6033535

SCHEMBL6033535

CCCCOC(=O)NC(C)N

nearest known ligand 0.50

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
HPGD P15428 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ACHE P22303 10/20 0.47
ALDH1A1 P00352 1/20 0.47
ATM Q13315 1/20 0.44
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8382659 0.84 EPHX1 (0.52) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL2551779 0.82 EPHX1 (0.50) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL27756824 0.82 EPHX1 (0.50) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL5128756 0.82 EPHX1 (0.50) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL29223070 0.81 EPHX1 (0.46) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL31440730 0.81 EPHX1 (0.46) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL7771457 0.81 EPHX1 (0.46) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL7786505 0.81 EPHX1 (0.46) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL1504664 0.81 SMN1; SMN2 (0.42) EPHX1SMN1; SMN2NPC1RAB9AHPGD
SCHEMBL7556363 0.81 RAB9A (0.51) EPHX1SMN1; SMN2NPC1RAB9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689789-A2 NOVEL CYCLODEXTRIN DIMERS AND DERIVATIVES THEREOF, METHODS FOR PREPARING THEM AND THEIR USE, IN PARTICULAR, FOR SOLUBILIZING PHARMACOLOGICALLY ACTIVE SUBSTANCES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2006-08-16 EP disclosed
WO-2005054303-A2 CYCLODEXTRIN DIMERS AND DERIVATIVES THEREOF, METHODS FOR PREPARING THEM AND THEIR USE, IN PARTICULAR, FOR SOLUBILIZING PHARMACOLOGICALLY ACTIVE SUBSTANCES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2005-06-16 WO disclosed
WO-2004101589-A1 NOVEL 14 AND 15 MEMBERED-RING COMPOUNDS GLAXO GROUP LIMITED (GB) 2004-11-25 WO disclosed
WO-1997043289-A1 LARGE SYNTHETIC COMPOUNDS BASED ON ELECTRON DONOR AND ELECTRON ACCEPTOR INTERACTIONS BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM (US) 1997-11-20 WO disclosed