SCHEMBL6045486

SCHEMBL6045486

c1ccc(CCNc2nc(Nc3cc(C4CC4)n[nH]3)c3ccccc3n2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.53
APP P05067 9/20 0.53
ACHE P22303 8/20 0.53
BCHE P06276 6/20 0.53
GRK6 P43250 2/20 0.52
AURKA O14965 1/20 0.52
NTRK1 P04629 2/20 0.51
IGF1R P08069 1/20 0.47
NTRK3 Q16288 1/20 0.46
NTRK2 Q16620 1/20 0.46
RAD52 P43351 1/20 0.45
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
MAPT P10636 1/20 0.44
PKM P14618 1/20 0.44
UBE2N P61088 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RCE1 Q9Y256 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2203633 0.94 NTRK1 (0.49) SLC2A1APPACHEBCHEGRK6
Benzene SCHEMBL27577366 0.86 BCHE (0.52) APPACHEBCHEGRK6NTRK1
SCHEMBL2206518 0.85 NTRK1 (0.51) APPACHEBCHENTRK1IGF1R
SCHEMBL2203233 0.85 NTRK1 (0.46) SLC2A1APPGRK6AURKANTRK1
SCHEMBL2205064 0.85 NTRK1 (0.46) APPACHEBCHEGRK6AURKA
SCHEMBL2204246 0.83 ULK1 (0.57) AURKANTRK1
SCHEMBL2200909 0.82 ULK1 (0.51) SLC2A1AURKANTRK1KDM4EALDH1A1
SCHEMBL2204494 0.82 ULK1 (0.51) GRK6AURKANTRK1
SCHEMBL11340376 0.82 IGF1R (0.70) NTRK1IGF1R
SCHEMBL12430677 0.82 NTRK1 (0.75) GRK6AURKANTRK1IGF1RNTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1345925-B1 PYRAZOLE COMPOUNDS USEFUL AS PROTEIN KINASE INHIBITORS VERTEX PHARMA (US) 2006-05-17 EP claimed