SCHEMBL6047580

SCHEMBL6047580

COc1ccc(C2=C(Cl)C(Cl)=CC[CH]2)c(-c2cccc([N+](=O)[O-])c2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
ALDH1A1 P00352 2/20 0.42
PKM P14618 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PLAU P00749 2/20 0.40
NFE2L2 Q16236 2/20 0.40
KEAP1 Q14145 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40
PLG P00747 1/20 0.40
PLAT P00750 1/20 0.40
MAOB P27338 1/20 0.38
HPGD P15428 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
CA14 Q9ULX7 1/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047578 0.85 CYP1A1 (0.42) ALDH1A1MAOB
SCHEMBL6047634 0.83 CYP1A1 (0.40) KMT2AMAOB
SCHEMBL6047612 0.82 MAOB (0.40) MAPTMEN1KMT2AALDH1A1NPSR1
SCHEMBL6047630 0.81 CYP3A4 (0.39) ALDH1A1MAOB
SCHEMBL6047641 0.76 ALKBH3 (0.34) MAPTMEN1KMT2AALDH1A1NPSR1
SCHEMBL6047590 0.75 MEN1 (0.41) MAPTMEN1KMT2AALDH1A1PKM
SCHEMBL6047654 0.74 NUDT1 (0.42) MAPTMEN1KMT2AALDH1A1HPGD
SCHEMBL28920300 0.73 NFE2L2 (0.51) MAPTMEN1KMT2AALDH1A1PKM
SCHEMBL30009634 0.73 NFE2L2 (0.51) MAPTMEN1KMT2AALDH1A1PKM
SCHEMBL6047586 0.73 CHRNA7 (0.35) MAPTMEN1KMT2ANPSR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed