SCHEMBL6047587

SCHEMBL6047587

FC(F)(F)C1=CC[CH]C(c2cccc(C(F)(F)F)c2)=C1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.42
KDM1A O60341 1/20 0.39
KIF11 P52732 1/20 0.38
NOTUM Q6P988 2/20 0.38
IDO1 P14902 1/20 0.38
ADORA2A P29274 2/20 0.38
ADORA1 P30542 2/20 0.38
ASIC3 Q9UHC3 1/20 0.38
SCN2A Q99250 2/20 0.37
MAOB P27338 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
GALR1 P47211 1/20 0.37
CTSS P25774 1/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047625 0.83 HTR2C (0.35) HTR2CNOTUMTSHRHTR1AHTR7
SCHEMBL1263144 0.71 TSHR (0.58) HTR2CKDM1AKIF11NOTUMIDO1
SCHEMBL29678302 0.71 TSHR (0.58) HTR2CKDM1AKIF11NOTUMIDO1
SCHEMBL17135818 0.70 HTR2C (0.43) HTR2CKDM1AKIF11NOTUMIDO1
Ammonia Solution, Strong SCHEMBL20472961 0.69 MAOB (0.56) HTR2CKDM1AKIF11NOTUMIDO1
SCHEMBL27895569 0.68 HTR2C (0.44) HTR2CKDM1AKIF11NOTUMIDO1
SCHEMBL6047584 0.68 MAPT (0.42) HTR2CKDM1ANOTUMIDO1ADORA2A
SCHEMBL1065756 0.66 HTR2C (0.53) HTR2CKDM1ANOTUMIDO1ASIC3
SCHEMBL1538783 0.66 MAOB (0.50) HTR2CKDM1AKIF11NOTUMIDO1
SCHEMBL29420699 0.66 KIF11 (0.62) KDM1AKIF11NOTUMIDO1ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed