SCHEMBL6047650

SCHEMBL6047650

COc1ccc(C2=C(Cl)C(Cl)=CC[CH]2)c(-c2ccccc2C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP24A1 Q07973 3/20 0.40
MAPK14 Q16539 1/20 0.39
CYP27A1 Q02318 1/20 0.37
TEK Q02763 1/20 0.37
CYP1A2 P05177 3/20 0.36
CYP3A4 P08684 3/20 0.36
ALOX15 P16050 3/20 0.36
CYP2C19 P33261 3/20 0.36
TSHR P16473 2/20 0.36
CYP2D6 P10635 2/20 0.36
USP2 O75604 1/20 0.36
TRPA1 O75762 2/20 0.36
TRPM8 Q7Z2W7 2/20 0.36
THRA P10827 1/20 0.36
THRB P10828 1/20 0.36
PDK2 Q15119 2/20 0.36
HSD11B1 P28845 2/20 0.35
MAPT P10636 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047654 0.80 NUDT1 (0.42) MAPK14CYP1A2CYP3A4ALOX15CYP2C19
SCHEMBL6047586 0.78 CHRNA7 (0.35) CYP1A2ALOX15CYP2C19CYP2D6MAPT
SCHEMBL6047628 0.76 ABL1 (0.47) TSHRMAPTNPC1RAB9ASMN1; SMN2
SCHEMBL6047634 0.75 CYP1A1 (0.40) MAPK14CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL6047641 0.75 ALKBH3 (0.34) CYP1A2CYP3A4ALOX15CYP2C19CYP2D6
SCHEMBL6047612 0.74 MAOB (0.40) MAPK14CYP1A2CYP3A4CYP2C19TSHR
SCHEMBL6047630 0.74 CYP3A4 (0.39) MAPK14CYP1A2CYP3A4CYP2C19CYP2D6
SCHEMBL6047622 0.73 CYP24A1 (0.40) CYP24A1MAPK14CYP27A1TEKCYP1A2
SCHEMBL6047638 0.66 MAPT (0.34) TSHRTHRBMAPTKDM4ENPC1
SCHEMBL31557643 0.65 CYP24A1 (0.49) CYP24A1MAPK14CYP27A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed