SCHEMBL6047622

SCHEMBL6047622

COc1ccc(C2=CC(Oc3ccccc3)=CC[CH]2)c(-c2ccccc2C(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP24A1 Q07973 2/20 0.40
CYP27A1 Q02318 1/20 0.40
MAPK14 Q16539 1/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PDK2 Q15119 2/20 0.37
THRA P10827 1/20 0.37
THRB P10828 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP1A2 P05177 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP3A4 P08684 2/20 0.35
ALOX15 P16050 2/20 0.35
TSHR P16473 2/20 0.35
USP2 O75604 1/20 0.35
CYP2D6 P10635 1/20 0.35
TRPA1 O75762 1/20 0.35
TRPM8 Q7Z2W7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047626 0.83 NPC1 (0.36) MAPTPDK2MEN1KMT2ACYP1A2
SCHEMBL6047656 0.82 HCRTR1 (0.36) PDK2
SCHEMBL6047648 0.81 NAAA (0.42) THRATHRBCYP1A2CYP2C19CYP3A4
SCHEMBL6047643 0.80 P2RX7 (0.37) MAPK14THRATHRBMEN1KMT2A
SCHEMBL6047659 0.80 THRA (0.39) THRATHRBAKR1C4AKR1C3AKR1C2
SCHEMBL6047633 0.79 PTPN1 (0.36) MAPTCYP1A2CYP2C19CYP3A4CYP2C9
SCHEMBL6047596 0.78 ABL1 (0.45) LMNAMAPTMEN1KMT2ACYP3A4
SCHEMBL6047600 0.77 ACHE (0.39) LMNAMAPTTDP1THRATHRB
SCHEMBL6047613 0.76 THRA (0.39) LMNAMAPTTHRATHRBCYP1A2
SCHEMBL6047602 0.76 NAAA (0.37) MAPK14MAPTTHRATHRBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed