SCHEMBL6047925

SCHEMBL6047925

Cc1cc2c(c(-c3cc(Cl)ccc3Cl)c1)OC(CN(C)N(C)CC1Cc3cc(C)cc(-c4cc(Cl)ccc4Cl)c3O1)C2

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AQP1 P29972 3/20 0.44
S1PR4 O95977 3/20 0.36
EZH2 Q15910 1/20 0.35
METAP1 P53582 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
TRPM4 Q8TD43 1/20 0.32
TRPM5 Q9NZQ8 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
RAPGEF4 Q8WZA2 1/20 0.30
IDO1 P14902 1/20 0.30
SIRT2 Q8IXJ6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047924 0.93 AQP1 (0.41) AQP1S1PR4EZH2HTR2AHTR2C
SCHEMBL4789302 0.88 AQP1 (0.45) AQP1S1PR4EZH2METAP1HRH4
SCHEMBL4231582 0.87 AQP1 (0.40) AQP1S1PR4EZH2METAP1KDM4E
SCHEMBL4831109 0.87 AQP1 (0.40) AQP1S1PR4EZH2METAP1KDM4E
SCHEMBL4220746 0.85 AQP1 (0.60) AQP1S1PR4EZH2HRH4HRH3
SCHEMBL6047906 0.83 AQP1 (0.37) AQP1EZH2METAP1TRPM5ALDH1A1
SCHEMBL4220767 0.83 AQP1 (0.64) AQP1S1PR4EZH2HRH4HRH3
SCHEMBL4220770 0.83 AQP1 (0.49) AQP1S1PR4EZH2HRH4HRH3
SCHEMBL4790052 0.83 AQP1 (0.44) AQP1S1PR4EZH2HRH4HRH3
SCHEMBL5142550 0.82 AQP1 (0.49) AQP1EZH2METAP1HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed