SCHEMBL6049009

SCHEMBL6049009

N=C(N)NC(N)CCCN

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
GSR P00390 1/20 0.31
DPP4 P27487 1/20 0.31
DPP8 Q6V1X1 1/20 0.31
DPP9 Q86TI2 1/20 0.31
DPP7 Q9UHL4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5670726 0.80 CA1 (0.38) DPP4DPP8DPP9DPP7
SCHEMBL28846838 0.79 CYP1A2 (0.34) CYP1A2CYP2C19
Hydrochloric Acid SCHEMBL28574831 0.77 OPRM1 (0.41) CYP1A2DPP7
SCHEMBL18434625 0.75 EPHX1 (0.32)
SCHEMBL7689323 0.75 HIF1A (0.33)
SCHEMBL349164 0.75 ENPEP (0.46) CYP1A2GSR
SCHEMBL23092019 0.74
SCHEMBL6048824 0.74
SCHEMBL3958831 0.74
Sulfuric Acid SCHEMBL12803038 0.71 TP53 (0.55) DPP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615946-A2 PROTEOLYTIC AND COVALENT ANTIBODIES The University of Texas (US) 2006-01-18 EP disclosed
EP-1610808-A2 COVALENT ATTACHMENT OF LIGANDS TO NUCLEOPHILIC PROTEINS GUIDED BY NON-COVALENT BINDING University of Texas Medical School (US) 2006-01-04 EP disclosed
WO-2004087735-A2 PROTEOLYTIC AND COVALENT ANTIBODIES THE UNIVERSITY OF TEXAS (US) 2004-10-14 WO disclosed
WO-2004087059-A2 COVALENT ATTACHMENT OF LIGANDS TO NUCLEOPHILIC PROTEINS GUIDED BY NON-COVALENT BINDING THE UNIVERSITY OF TEXAS (US) 2004-10-14 WO disclosed