SCHEMBL6049129

SCHEMBL6049129

N#Cc1cc(CCBr)cc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.43
RXRG P48443 1/20 0.43
MRGPRX4 Q96LA9 4/20 0.40
KIF11 P52732 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
XDH P47989 1/20 0.36
TAS2R14 Q9NYV8 1/20 0.35
IDO1 P14902 2/20 0.34
DAO P14920 1/20 0.33
TACR1 P25103 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
ENPP2 Q13822 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL130428 0.86 RXRA (0.46) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL29812995 0.86 RXRA (0.46) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL2393670 0.81 IDO1 (0.48) RXRARXRGIDO1DAOTACR1
SCHEMBL17319636 0.80 RXRA (0.47) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL24108532 0.79 RXRA (0.46) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL2390020 0.79 RXRA (0.49) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL172834 0.79 RXRA (0.46) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL129227 0.79 RXRA (0.49) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL169517 0.79 RXRA (0.46) RXRARXRGMRGPRX4KIF11L3MBTL1
SCHEMBL172532 0.79 RXRA (0.46) RXRARXRGMRGPRX4KIF11L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008355-A Azaindole derivatives as protein kinase inhibitors ORIBASE PHARMA 2015-10-28 CN disclosed
CN-103172562-B Trisubstituted amine compounds as inhibitors of cholesteryl ester transfer protein CETP TANABE SEIYAKU CO 2015-04-22 CN disclosed
CN-101374817-B Trisubstituted amine compounds as inhibitors of cholesteryl ester transfer protein CETP MITSUBISHI TANABE PHARMA CORP 2014-07-30 CN disclosed
CN-103172562-A Trisubstituted amine compounds as inhibitors of cholesteryl ester transfer protein CETP TANABE SEIYAKU CO 2013-06-26 CN disclosed
CN-101466679-A Process for preparing tetrahydroquinoline derivatives MITSUBISHI TANABE PHARMA CORP (JP) 2009-06-24 CN disclosed
CN-101437804-A Dibenzyl amine compounds and derivatives PFIZER PROD INC (US) 2009-05-20 CN disclosed
CN-101374817-A Trisubstituted amine compounds as inhibitors of cholesteryl ester transfer protein CETP MITSUBISHI TANABE PHARMA CORP (JP) 2009-02-25 CN disclosed
CN-1289467-C Dibenzylamine compound and pharmaceutical use thereof JAPAN TOBACCO INC (JP) 2006-12-13 CN disclosed
JP-2006045095-A 3-FORMYL-5-TRIFLUOROMETHYLBENZONITRILE DERIVATIVE AND METHOD FOR PRODUCING THE SAME CENTRAL GLASS CO LTD 2006-02-16 JP disclosed
CN-1617850-A Dibenzylamine compound and medicinal use thereof JAPAN TOBACCO INC (JP) 2005-05-18 CN disclosed